3-Isoquinolinecarboxylic acid, 1,2,3,4-tetrahydro-2-(5-((aminoiminomethyl)amino)-2-(((6,7-dimethoxy-2-naphthalenyl)sulfonyl)amino)-1-oxopentyl)- structure

3-Isoquinolinecarboxylic acid, 1,2,3,4-tetrahydro-2-(5-((aminoiminomethyl)amino)-2-(((6,7-dimethoxy-2-naphthalenyl)sulfonyl)amino)-1-oxopentyl)-

TL;DR: 3-Isoquinolinecarboxylic acid, 1,2,3,4-tetrahydro-2-(5-((aminoiminomethyl)amino)-2-(((6,7-dimethoxy-2-naphthalenyl)sulfonyl)amino)-1-oxopentyl)- (CAS 66937-37-9) is a chemical compound with molecular formula C28H33N5O7S and molecular weight 583.21 g/mol, supplied by Kehong Biological (Henan Kehong Biological Technology Co., Ltd.) with CRO/CDMO custom synthesis services.

2-[5-(diaminomethylideneamino)-2-[(6,7-dimethoxynaphthalen-2-yl)sulfonylamino]pentanoyl]-3,4-dihydro-1H-isoquinoline-3-carboxylic acid

Also Known As: 3-Isoquinolinecarboxylic acid, 1,2,3,4-tetrahydro-2-(5-((aminoiminomethyl)amino)-2-(((6,7-dimethoxy-2-naphthalenyl)sulfonyl)amino)-1-oxopentyl)-, 2-[5-(diaminomethylideneamino)-2-[(6,7-dimethoxynaphthalen-2-yl)sulfonylamino]pentanoyl]-3,4-dihydro-1H-isoquinoline-3-carboxylic acid, 2-[N~2~-(6,7-Dimethoxynaphthalene-2-sulfonyl)arginyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid, RefChem:280173

CAS: 66937-37-9
Molecular Formula C28H33N5O7S
Molecular Weight 583.21 g/mol
LogP 1.5956
Topological Polar Surface Area 186.64 Ų
Hydrogen Bond Donors 4
Hydrogen Bond Acceptors 7
Rotatable Bonds 11
Exact Mass 583.2101
Heavy Atoms 41
Complexity 1587.9419

Chemical Identifiers

CAS Number 66937-37-9
SMILES COC1=C(C=C2C=C(C=CC2=C1)S(=O)(=O)NC(CCCN=C(N)N)C(=O)N3CC4=CC=CC=C4CC3C(=O)O)OC

Product Overview

3-Isoquinolinecarboxylic acid, 1,2,3,4-tetrahydro-2-(5-((aminoiminomethyl)amino)-2-(((6,7-dimethoxy-2-naphthalenyl)sulfonyl)amino)-1-oxopentyl)- (CAS 66937-37-9), with molecular formula C28H33N5O7S and molecular weight 583.21 g/mol. IUPAC: 2-[5-(diaminomethylideneamino)-2-[(6,7-dimethoxynaphthalen-2-yl)sulfonylamino]pentanoyl]-3,4-dihydro-1H-isoquinoline-3-carboxylic acid.

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Safety Data Sheet (MSDS / SDS) View the Laboratory Chemical Safety Summary (LCSS) on PubChem — includes GHS classifications, hazard statements, first aid measures, and handling precautions.
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Chemical Property Profile of 3-Isoquinolinecarboxylic acid, 1,2,3,4-tetrahydro-2-(5-((aminoiminomethyl)amino)-2-(((6,7-dimethoxy-2-naphthalenyl)sulfonyl)amino)-1-oxopentyl)-

XLogP
1.5956
TPSA (Topological Polar Surface Area)
186.64
Hydrogen Bond Donors
4
Hydrogen Bond Acceptors
7
Rotatable Bonds
11
Heavy Atoms
41
Complexity
1587.9419
Exact Mass
583.2101
Monoisotopic Mass
583.2101
Data Source: Chemical property values are referenced from PubChem, the world's largest open chemistry database maintained by the National Center for Biotechnology Information (NCBI), U.S. National Library of Medicine.

Property Insights of 3-Isoquinolinecarboxylic acid, 1,2,3,4-tetrahydro-2-(5-((aminoiminomethyl)amino)-2-(((6,7-dimethoxy-2-naphthalenyl)sulfonyl)amino)-1-oxopentyl)-

The XLogP value of 1.5956 suggests moderate lipophilicity, balancing water solubility and membrane permeability for 3-Isoquinolinecarboxylic acid, 1,2,3,4-tetrahydro-2-(5-((aminoiminomethyl)amino)-2-(((6,7-dimethoxy-2-naphthalenyl)sulfonyl)amino)-1-oxopentyl)-. The TPSA of 186.64 Ų indicates high polarity, suggesting 3-Isoquinolinecarboxylic acid, 1,2,3,4-tetrahydro-2-(5-((aminoiminomethyl)amino)-2-(((6,7-dimethoxy-2-naphthalenyl)sulfonyl)amino)-1-oxopentyl)- may have limited membrane permeability but good aqueous solubility. Following Lipinski's Rule of Five, 3-Isoquinolinecarboxylic acid, 1,2,3,4-tetrahydro-2-(5-((aminoiminomethyl)amino)-2-(((6,7-dimethoxy-2-naphthalenyl)sulfonyl)amino)-1-oxopentyl)- has 4 hydrogen bond donor(s) and 7 hydrogen bond acceptor(s), which may warrant consideration for formulation optimization.

Frequently Asked Questions

What is the typical lead time for this product?
Lead time typically ranges from 3-7 business days for in-stock items. For larger quantities or custom orders, please contact us for specific lead times.
Can you provide samples for testing?
Yes, we offer sample quantities for quality testing. Please submit an inquiry with your requirements and we will arrange samples accordingly.
What documentation do you provide with the product?
We provide COA (Certificate of Analysis), MSDS (Material Safety Data Sheet), and technical data sheets with each shipment.
Do you ship internationally?
Yes, we ship to most countries worldwide. Shipping costs and delivery times vary by location. Please contact us for specific shipping information.

Frequently Asked Questions

What is the CAS number of 3-Isoquinolinecarboxylic acid, 1,2,3,4-tetrahydro-2-(5-((aminoiminomethyl)amino)-2-(((6,7-dimethoxy-2-naphthalenyl)sulfonyl)amino)-1-oxopentyl)-?

The CAS number of 3-Isoquinolinecarboxylic acid, 1,2,3,4-tetrahydro-2-(5-((aminoiminomethyl)amino)-2-(((6,7-dimethoxy-2-naphthalenyl)sulfonyl)amino)-1-oxopentyl)- is 66937-37-9.

What is the molecular formula of 3-Isoquinolinecarboxylic acid, 1,2,3,4-tetrahydro-2-(5-((aminoiminomethyl)amino)-2-(((6,7-dimethoxy-2-naphthalenyl)sulfonyl)amino)-1-oxopentyl)-?

The molecular formula of 3-Isoquinolinecarboxylic acid, 1,2,3,4-tetrahydro-2-(5-((aminoiminomethyl)amino)-2-(((6,7-dimethoxy-2-naphthalenyl)sulfonyl)amino)-1-oxopentyl)- is C28H33N5O7S.

What is the molecular weight of 3-Isoquinolinecarboxylic acid, 1,2,3,4-tetrahydro-2-(5-((aminoiminomethyl)amino)-2-(((6,7-dimethoxy-2-naphthalenyl)sulfonyl)amino)-1-oxopentyl)-?

The molecular weight of 3-Isoquinolinecarboxylic acid, 1,2,3,4-tetrahydro-2-(5-((aminoiminomethyl)amino)-2-(((6,7-dimethoxy-2-naphthalenyl)sulfonyl)amino)-1-oxopentyl)- is 583.21 g/mol.

Where can I buy 3-Isoquinolinecarboxylic acid, 1,2,3,4-tetrahydro-2-(5-((aminoiminomethyl)amino)-2-(((6,7-dimethoxy-2-naphthalenyl)sulfonyl)amino)-1-oxopentyl)-?

You can request a quote for 3-Isoquinolinecarboxylic acid, 1,2,3,4-tetrahydro-2-(5-((aminoiminomethyl)amino)-2-(((6,7-dimethoxy-2-naphthalenyl)sulfonyl)amino)-1-oxopentyl)- directly from KEHONG BIO. Contact us or email info@kehongbio.com for pricing and availability.

Does KEHONG BIO offer custom synthesis for 3-Isoquinolinecarboxylic acid, 1,2,3,4-tetrahydro-2-(5-((aminoiminomethyl)amino)-2-(((6,7-dimethoxy-2-naphthalenyl)sulfonyl)amino)-1-oxopentyl)-?

Yes, KEHONG BIO provides custom synthesis services for 3-Isoquinolinecarboxylic acid, 1,2,3,4-tetrahydro-2-(5-((aminoiminomethyl)amino)-2-(((6,7-dimethoxy-2-naphthalenyl)sulfonyl)amino)-1-oxopentyl)- and related compounds. Contact us with your specific requirements including quantity, purity, and timeline.

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