N1-(2-morpholinoquinazolin-4-yl)-N3-(2-nitro-4-(trifluoromethyl)phenyl)propane-1,3-diamine structure

N1-(2-morpholinoquinazolin-4-yl)-N3-(2-nitro-4-(trifluoromethyl)phenyl)propane-1,3-diamine

TL;DR: N1-(2-morpholinoquinazolin-4-yl)-N3-(2-nitro-4-(trifluoromethyl)phenyl)propane-1,3-diamine (CAS 597545-76-1) is a chemical compound with molecular formula C22H23F3N6O3 and molecular weight 476.18 g/mol, supplied by Kehong Biological (Henan Kehong Biological Technology Co., Ltd.) with CRO/CDMO custom synthesis services.

N'-(2-morpholin-4-ylquinazolin-4-yl)-N-[2-nitro-4-(trifluoromethyl)phenyl]propane-1,3-diamine

Also Known As: N1-(2-morpholinoquinazolin-4-yl)-N3-(2-nitro-4-(trifluoromethyl)phenyl)propane-1,3-diamine, N'-(2-morpholin-4-ylquinazolin-4-yl)-N-[2-nitro-4-(trifluoromethyl)phenyl]propane-1,3-diamine, N-(2-morpholin-4-ylquinazolin-4-yl)-N'-[2-nitro-4-(trifluoromethyl)phenyl]propane-1,3-diamine, N-(2-MORPHOLINO-4-QUINAZOLINYL)-N-{3-[2-NITRO-4-(TRIFLUOROMETHYL)ANILINO]PROPYL}AMINE, N-[2-(4-morpholinyl)-4-quinazolinyl]-N'-[2-nitro-4-(trifluoromethyl)phenyl]-1,3-propanediamine

CAS: 597545-76-1
Molecular Formula C22H23F3N6O3
Molecular Weight 476.18 g/mol
LogP 4.3075
Topological Polar Surface Area 105.45 Ų
Hydrogen Bond Donors 2
Hydrogen Bond Acceptors 8
Rotatable Bonds 8
Exact Mass 476.17838
Heavy Atoms 34
Complexity 1168.3204

Chemical Identifiers

CAS Number 597545-76-1
SMILES C1COCCN1C2=NC3=CC=CC=C3C(=N2)NCCCNC4=C(C=C(C=C4)C(F)(F)F)[N+](=O)[O-]

Product Overview

N1-(2-morpholinoquinazolin-4-yl)-N3-(2-nitro-4-(trifluoromethyl)phenyl)propane-1,3-diamine (CAS 597545-76-1), with molecular formula C22H23F3N6O3 and molecular weight 476.18 g/mol. IUPAC: N'-(2-morpholin-4-ylquinazolin-4-yl)-N-[2-nitro-4-(trifluoromethyl)phenyl]propane-1,3-diamine.

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Safety Data Sheet (MSDS / SDS) View the Laboratory Chemical Safety Summary (LCSS) on PubChem — includes GHS classifications, hazard statements, first aid measures, and handling precautions.
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Chemical Property Profile of N1-(2-morpholinoquinazolin-4-yl)-N3-(2-nitro-4-(trifluoromethyl)phenyl)propane-1,3-diamine

XLogP
4.3075
TPSA (Topological Polar Surface Area)
105.45
Hydrogen Bond Donors
2
Hydrogen Bond Acceptors
8
Rotatable Bonds
8
Heavy Atoms
34
Complexity
1168.3204
Exact Mass
476.17838
Monoisotopic Mass
476.17838
Data Source: Chemical property values are referenced from PubChem, the world's largest open chemistry database maintained by the National Center for Biotechnology Information (NCBI), U.S. National Library of Medicine.

Property Insights of N1-(2-morpholinoquinazolin-4-yl)-N3-(2-nitro-4-(trifluoromethyl)phenyl)propane-1,3-diamine

The XLogP value of 4.3075 indicates that N1-(2-morpholinoquinazolin-4-yl)-N3-(2-nitro-4-(trifluoromethyl)phenyl)propane-1,3-diamine is lipophilic (fat-soluble), which may influence its absorption, distribution, and formulation strategy. The TPSA of 105.45 Ų falls within the moderate polarity range, balancing permeability and solubility for N1-(2-morpholinoquinazolin-4-yl)-N3-(2-nitro-4-(trifluoromethyl)phenyl)propane-1,3-diamine. Following Lipinski's Rule of Five, N1-(2-morpholinoquinazolin-4-yl)-N3-(2-nitro-4-(trifluoromethyl)phenyl)propane-1,3-diamine has 2 hydrogen bond donor(s) and 8 hydrogen bond acceptor(s), all within the drug-like range, suggesting favorable oral bioavailability potential.

Frequently Asked Questions

What is the typical lead time for this product?
Lead time typically ranges from 3-7 business days for in-stock items. For larger quantities or custom orders, please contact us for specific lead times.
Can you provide samples for testing?
Yes, we offer sample quantities for quality testing. Please submit an inquiry with your requirements and we will arrange samples accordingly.
What documentation do you provide with the product?
We provide COA (Certificate of Analysis), MSDS (Material Safety Data Sheet), and technical data sheets with each shipment.
Do you ship internationally?
Yes, we ship to most countries worldwide. Shipping costs and delivery times vary by location. Please contact us for specific shipping information.

Frequently Asked Questions

What is the CAS number of N1-(2-morpholinoquinazolin-4-yl)-N3-(2-nitro-4-(trifluoromethyl)phenyl)propane-1,3-diamine?

The CAS number of N1-(2-morpholinoquinazolin-4-yl)-N3-(2-nitro-4-(trifluoromethyl)phenyl)propane-1,3-diamine is 597545-76-1.

What is the molecular formula of N1-(2-morpholinoquinazolin-4-yl)-N3-(2-nitro-4-(trifluoromethyl)phenyl)propane-1,3-diamine?

The molecular formula of N1-(2-morpholinoquinazolin-4-yl)-N3-(2-nitro-4-(trifluoromethyl)phenyl)propane-1,3-diamine is C22H23F3N6O3.

What is the molecular weight of N1-(2-morpholinoquinazolin-4-yl)-N3-(2-nitro-4-(trifluoromethyl)phenyl)propane-1,3-diamine?

The molecular weight of N1-(2-morpholinoquinazolin-4-yl)-N3-(2-nitro-4-(trifluoromethyl)phenyl)propane-1,3-diamine is 476.18 g/mol.

Where can I buy N1-(2-morpholinoquinazolin-4-yl)-N3-(2-nitro-4-(trifluoromethyl)phenyl)propane-1,3-diamine?

You can request a quote for N1-(2-morpholinoquinazolin-4-yl)-N3-(2-nitro-4-(trifluoromethyl)phenyl)propane-1,3-diamine directly from KEHONG BIO. Contact us or email info@kehongbio.com for pricing and availability.

Does KEHONG BIO offer custom synthesis for N1-(2-morpholinoquinazolin-4-yl)-N3-(2-nitro-4-(trifluoromethyl)phenyl)propane-1,3-diamine?

Yes, KEHONG BIO provides custom synthesis services for N1-(2-morpholinoquinazolin-4-yl)-N3-(2-nitro-4-(trifluoromethyl)phenyl)propane-1,3-diamine and related compounds. Contact us with your specific requirements including quantity, purity, and timeline.

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