E 4018 structure

E 4018

TL;DR: E 4018 (CAS 251375-82-3) is a chemical compound with molecular formula C21H29N3O8 and molecular weight 451.20 g/mol, supplied by Kehong Biological (Henan Kehong Biological Technology Co., Ltd.) with CRO/CDMO custom synthesis services.

E 4018

N,N-dimethyl-2-[(2-methylpyrazol-3-yl)-phenylmethoxy]ethanamine;2-hydroxypropane-1,2,3-tricarboxylic acid

Also Known As: Cizolirtine citrate, null, E-3710 citrate, Cizolirtine citrate [MI], 251375-82-3 (citrate)

CAS: 251375-82-3
Molecular Formula C21H29N3O8
Molecular Weight 451.20 g/mol
LogP 0.8392
Topological Polar Surface Area 162.0 Ų
Hydrogen Bond Donors 4
Hydrogen Bond Acceptors 10
Rotatable Bonds 11
Exact Mass 451.19547
Heavy Atoms 32
Complexity 481.0

Chemical Identifiers

CAS Number 251375-82-3
SMILES CN1C(=CC=N1)C(C2=CC=CC=C2)OCCN(C)C.C(C(=O)O)C(CC(=O)O)(C(=O)O)O
InChIKey JLKUMSHHQYQLSG-UHFFFAOYSA-N

Patent-Derived Application Labels

Derived from 3 IPC patent classification(s) across the SureChEMBL global patent database.

Heterocyclic Building Blocks (18 patents) Organic Building Blocks (3 patents) Pharmaceutical Intermediates (94 patents)

Product Overview

E 4018 (CAS 251375-82-3), with molecular formula C21H29N3O8 and molecular weight 451.20 g/mol. IUPAC: N,N-dimethyl-2-[(2-methylpyrazol-3-yl)-phenylmethoxy]ethanamine;2-hydroxypropane-1,2,3-tricarboxylic acid.

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Safety Data Sheet (MSDS / SDS) View the Laboratory Chemical Safety Summary (LCSS) on PubChem — includes GHS classifications, hazard statements, first aid measures, and handling precautions.
View MSDS →

Chemical Property Profile of E 4018

XLogP
0.8392
TPSA (Topological Polar Surface Area)
162.0
Hydrogen Bond Donors
4
Hydrogen Bond Acceptors
10
Rotatable Bonds
11
Heavy Atoms
32
Complexity
481.0
Exact Mass
451.19547
Monoisotopic Mass
451.19547
Data Source: Chemical property values are referenced from PubChem, the world's largest open chemistry database maintained by the National Center for Biotechnology Information (NCBI), U.S. National Library of Medicine.

Property Insights of E 4018

The XLogP value of 0.8392 suggests moderate lipophilicity, balancing water solubility and membrane permeability for E 4018. The TPSA of 162.0 Ų indicates high polarity, suggesting E 4018 may have limited membrane permeability but good aqueous solubility. Following Lipinski's Rule of Five, E 4018 has 4 hydrogen bond donor(s) and 10 hydrogen bond acceptor(s), all within the drug-like range, suggesting favorable oral bioavailability potential.

Frequently Asked Questions

What is the typical lead time for this product?
Lead time typically ranges from 3-7 business days for in-stock items. For larger quantities or custom orders, please contact us for specific lead times.
Can you provide samples for testing?
Yes, we offer sample quantities for quality testing. Please submit an inquiry with your requirements and we will arrange samples accordingly.
What documentation do you provide with the product?
We provide COA (Certificate of Analysis), MSDS (Material Safety Data Sheet), and technical data sheets with each shipment.
Do you ship internationally?
Yes, we ship to most countries worldwide. Shipping costs and delivery times vary by location. Please contact us for specific shipping information.

Frequently Asked Questions

What is the CAS number of E 4018?

The CAS number of E 4018 is 251375-82-3.

What is the molecular formula of E 4018?

The molecular formula of E 4018 is C21H29N3O8.

What is the molecular weight of E 4018?

The molecular weight of E 4018 is 451.20 g/mol.

Where can I buy E 4018?

You can request a quote for E 4018 directly from KEHONG BIO. Contact us or email info@kehongbio.com for pricing and availability.

Does KEHONG BIO offer custom synthesis for E 4018?

Yes, KEHONG BIO provides custom synthesis services for E 4018 and related compounds. Contact us with your specific requirements including quantity, purity, and timeline.

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