Clotiapine structure

Clotiapine

TL;DR: Clotiapine (CAS 2058-52-8) is a chemical compound with molecular formula C18H18ClN3S and molecular weight 343.09 g/mol, supplied by Kehong Biological (Henan Kehong Biological Technology Co., Ltd.) with CRO/CDMO custom synthesis services.

8-chloro-6-(4-methylpiperazin-1-yl)benzo[b][1,4]benzothiazepine

Also Known As: Clothiapine, Clotiapine, Entumin, Entumine, Etumine

CAS: 2058-52-8
Molecular Formula C18H18ClN3S
Molecular Weight 343.09 g/mol
LogP 3.6
Topological Polar Surface Area 44.1 Ų
Hydrogen Bond Donors 0
Hydrogen Bond Acceptors 3
Rotatable Bonds 1
Exact Mass 343.091
Heavy Atoms 23
Complexity 450.0

Chemical Identifiers

CAS Number 2058-52-8
SMILES CN1CCN(CC1)C2=NC3=CC=CC=C3SC4=C2C=C(C=C4)Cl
InChIKey KAAZGXDPUNNEFN-UHFFFAOYSA-N

Patent-Derived Application Labels

Derived from 10 IPC patent classification(s) across the SureChEMBL global patent database.

Agrochemicals (3 patents) Analytical Reagents (3 patents) Biotechnology (13 patents) Electronic Chemicals (4 patents) Heterocyclic Building Blocks (79 patents) +5 more

Product Overview

Clotiapine (CAS 2058-52-8), with molecular formula C18H18ClN3S and molecular weight 343.09 g/mol. IUPAC: 8-chloro-6-(4-methylpiperazin-1-yl)benzo[b][1,4]benzothiazepine.

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Safety Data Sheet (MSDS / SDS) View the Laboratory Chemical Safety Summary (LCSS) on PubChem — includes GHS classifications, hazard statements, first aid measures, and handling precautions.
View MSDS →

Chemical Property Profile of Clotiapine

XLogP
3.6
TPSA (Topological Polar Surface Area)
44.1
Hydrogen Bond Donors
0
Hydrogen Bond Acceptors
3
Rotatable Bonds
1
Heavy Atoms
23
Complexity
450.0
Exact Mass
343.091
Monoisotopic Mass
343.091
Data Source: Chemical property values are referenced from PubChem, the world's largest open chemistry database maintained by the National Center for Biotechnology Information (NCBI), U.S. National Library of Medicine.

Property Insights of Clotiapine

The XLogP value of 3.6 indicates that Clotiapine is lipophilic (fat-soluble), which may influence its absorption, distribution, and formulation strategy. With a topological polar surface area (TPSA) of 44.1 Ų, Clotiapine exhibits relatively low polarity, potentially indicating favorable cell membrane permeability. Following Lipinski's Rule of Five, Clotiapine has 0 hydrogen bond donor(s) and 3 hydrogen bond acceptor(s), all within the drug-like range, suggesting favorable oral bioavailability potential.

Frequently Asked Questions

What is the typical lead time for this product?
Lead time typically ranges from 3-7 business days for in-stock items. For larger quantities or custom orders, please contact us for specific lead times.
Can you provide samples for testing?
Yes, we offer sample quantities for quality testing. Please submit an inquiry with your requirements and we will arrange samples accordingly.
What documentation do you provide with the product?
We provide COA (Certificate of Analysis), MSDS (Material Safety Data Sheet), and technical data sheets with each shipment.
Do you ship internationally?
Yes, we ship to most countries worldwide. Shipping costs and delivery times vary by location. Please contact us for specific shipping information.

Frequently Asked Questions

What is the CAS number of Clotiapine?

The CAS number of Clotiapine is 2058-52-8.

What is the molecular formula of Clotiapine?

The molecular formula of Clotiapine is C18H18ClN3S.

What is the molecular weight of Clotiapine?

The molecular weight of Clotiapine is 343.09 g/mol.

Where can I buy Clotiapine?

You can request a quote for Clotiapine directly from KEHONG BIO. Contact us or email info@kehongbio.com for pricing and availability.

Does KEHONG BIO offer custom synthesis for Clotiapine?

Yes, KEHONG BIO provides custom synthesis services for Clotiapine and related compounds. Contact us with your specific requirements including quantity, purity, and timeline.

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