Aprosulate Sodium structure

Aprosulate Sodium

TL;DR: Aprosulate Sodium (CAS 123072-45-7) is a chemical compound with molecular formula C27H34N2Na16O70S16 and molecular weight 2385.31 g/mol, supplied by Kehong Biological (Henan Kehong Biological Technology Co., Ltd.) with CRO/CDMO custom synthesis services.

hexadecasodium;[(1S,2R,3R)-1-[(1R)-2-oxo-1-sulfonatooxy-2-[3-[[(2R,3S,4R,5R)-2,3,5,6-tetrasulfonatooxy-4-[(2S,3R,4S,5S,6R)-3,4,5-trisulfonatooxy-6-(sulfonatooxymethyl)oxan-2-yl]oxyhexanoyl]amino]propylamino]ethyl]-3,4-disulfonatooxy-2-[(2S,3R,4S,5S,6R)-3,4,5-trisulfonatooxy-6-(sulfonatooxymethyl)oxan-2-yl]oxybutyl] sulfate

Also Known As: Aprosulate Sodium, Aprosulate, Aprosulate sodique, Aprosulato sodico, Aprosulatum natricum

CAS: 123072-45-7
Molecular Formula C27H34N2Na16O70S16
Molecular Weight 2385.31 g/mol
LogP -68.05
Topological Polar Surface Area 1290.0 Ų
Hydrogen Bond Donors 2
Hydrogen Bond Acceptors 70
Rotatable Bonds 36
Exact Mass 2385.3057
Heavy Atoms 131
Complexity 4720.0

Chemical Identifiers

CAS Number 123072-45-7
SMILES C(CNC(=O)[C@@H]([C@H]([C@@H]([C@@H](COS(=O)(=O)[O-])OS(=O)(=O)[O-])O[C@H]1[C@@H]([C@H]([C@H]([C@H](O1)COS(=O)(=O)[O-])OS(=O)(=O)[O-])OS(=O)(=O)[O-])OS(=O)(=O)[O-])OS(=O)(=O)[O-])OS(=O)(=O)[O-])CNC(=O)[C@@H]([C@H]([C@@H]([C@@H](COS(=O)(=O)[O-])OS(=O)(=O)[O-])O[C@H]2[C@@H]([C@H]([C@H]([C@H](O2)COS(=O)(=O)[O-])OS(=O)(=O)[O-])OS(=O)(=O)[O-])OS(=O)(=O)[O-])OS(=O)(=O)[O-])OS(=O)(=O)[O-].[Na+].[Na+].[Na+].[Na+].[Na+].[Na+].[Na+].[Na+].[Na+].[Na+].[Na+].[Na+].[Na+].[Na+].[Na+].[Na+]
InChIKey CXKOATPJKFZCEL-HPXJARCXSA-A

Patent-Derived Application Labels

Derived from 3 IPC patent classification(s) across the SureChEMBL global patent database.

Analytical Reagents (2 patents) Biotechnology (2 patents) Pharmaceutical Intermediates (23 patents)

Product Overview

Aprosulate Sodium (CAS 123072-45-7), with molecular formula C27H34N2Na16O70S16 and molecular weight 2385.31 g/mol. IUPAC: hexadecasodium;[(1S,2R,3R)-1-[(1R)-2-oxo-1-sulfonatooxy-2-[3-[[(2R,3S,4R,5R)-2,3,5,6-tetrasulfonatooxy-4-[(2S,3R,4S,5S,6R)-3,4,5-trisulfonatooxy-6-(sulfonatooxymethyl)oxan-2-yl]oxyhexanoyl]amino]propylamino]ethyl]-3,4-disulfonatooxy-2-[(2S,3R,4S,5S,6R)-3,4,5-trisulfonatooxy-6-(sulfonatooxymethyl)oxan-2-yl]oxybutyl] sulfate.

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Safety Data Sheet (MSDS / SDS) View the Laboratory Chemical Safety Summary (LCSS) on PubChem — includes GHS classifications, hazard statements, first aid measures, and handling precautions.
View MSDS →

Chemical Property Profile of Aprosulate Sodium

XLogP
-68.05
TPSA (Topological Polar Surface Area)
1290.0
Hydrogen Bond Donors
2
Hydrogen Bond Acceptors
70
Rotatable Bonds
36
Heavy Atoms
131
Complexity
4720.0
Exact Mass
2385.3057
Monoisotopic Mass
2385.3057
Data Source: Chemical property values are referenced from PubChem, the world's largest open chemistry database maintained by the National Center for Biotechnology Information (NCBI), U.S. National Library of Medicine.

Property Insights of Aprosulate Sodium

The XLogP value of -68.05 indicates that Aprosulate Sodium is hydrophilic (water-soluble), making it suitable for aqueous formulations and biological assay applications. The TPSA of 1290.0 Ų indicates high polarity, suggesting Aprosulate Sodium may have limited membrane permeability but good aqueous solubility. Following Lipinski's Rule of Five, Aprosulate Sodium has 2 hydrogen bond donor(s) and 70 hydrogen bond acceptor(s), which may warrant consideration for formulation optimization.

Frequently Asked Questions

What is the typical lead time for this product?
Lead time typically ranges from 3-7 business days for in-stock items. For larger quantities or custom orders, please contact us for specific lead times.
Can you provide samples for testing?
Yes, we offer sample quantities for quality testing. Please submit an inquiry with your requirements and we will arrange samples accordingly.
What documentation do you provide with the product?
We provide COA (Certificate of Analysis), MSDS (Material Safety Data Sheet), and technical data sheets with each shipment.
Do you ship internationally?
Yes, we ship to most countries worldwide. Shipping costs and delivery times vary by location. Please contact us for specific shipping information.

Frequently Asked Questions

What is the CAS number of Aprosulate Sodium?

The CAS number of Aprosulate Sodium is 123072-45-7.

What is the molecular formula of Aprosulate Sodium?

The molecular formula of Aprosulate Sodium is C27H34N2Na16O70S16.

What is the molecular weight of Aprosulate Sodium?

The molecular weight of Aprosulate Sodium is 2385.31 g/mol.

Where can I buy Aprosulate Sodium?

You can request a quote for Aprosulate Sodium directly from KEHONG BIO. Contact us or email info@kehongbio.com for pricing and availability.

Does KEHONG BIO offer custom synthesis for Aprosulate Sodium?

Yes, KEHONG BIO provides custom synthesis services for Aprosulate Sodium and related compounds. Contact us with your specific requirements including quantity, purity, and timeline.

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