2,5-Dioxopyrrolidin-1-yl 1-(tert-butoxycarbonyl)prolinate structure

2,5-Dioxopyrrolidin-1-yl 1-(tert-butoxycarbonyl)prolinate

TL;DR: 2,5-Dioxopyrrolidin-1-yl 1-(tert-butoxycarbonyl)prolinate (CAS 102185-34-2) is a chemical compound with molecular formula C14H20N2O6 and molecular weight 312.13 g/mol, supplied by Kehong Biological (Henan Kehong Biological Technology Co., Ltd.) with CRO/CDMO custom synthesis services.

1-O-tert-butyl 2-O-(2,5-dioxopyrrolidin-1-yl) pyrrolidine-1,2-dicarboxylate

Also Known As: Boc-D-Pro-OSu, Boc-Pro-OSu, Boc-L-Pro-OSu, Boc-L-proline N-hydroxysuccinimide ester, BAS 00615791

CAS: 102185-34-2
Molecular Formula C14H20N2O6
Molecular Weight 312.13 g/mol
LogP 0.7
Topological Polar Surface Area 93.2 Ų
Hydrogen Bond Donors 0
Hydrogen Bond Acceptors 6
Rotatable Bonds 5
Exact Mass 312.13214
Heavy Atoms 22
Complexity 494.0

Chemical Identifiers

CAS Number 102185-34-2
SMILES CC(C)(C)OC(=O)N1CCCC1C(=O)ON2C(=O)CCC2=O
InChIKey DICWIJISMKZDDY-UHFFFAOYSA-N

Patent-Derived Application Labels

Derived from 2 IPC patent classification(s) across the SureChEMBL global patent database.

Heterocyclic Building Blocks (1 patents) Pharmaceutical Intermediates (4 patents)

Product Overview

2,5-Dioxopyrrolidin-1-yl 1-(tert-butoxycarbonyl)prolinate (CAS 102185-34-2), with molecular formula C14H20N2O6 and molecular weight 312.13 g/mol. IUPAC: 1-O-tert-butyl 2-O-(2,5-dioxopyrrolidin-1-yl) pyrrolidine-1,2-dicarboxylate.

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Safety Data Sheet (MSDS / SDS) View the Laboratory Chemical Safety Summary (LCSS) on PubChem — includes GHS classifications, hazard statements, first aid measures, and handling precautions.
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Chemical Property Profile of 2,5-Dioxopyrrolidin-1-yl 1-(tert-butoxycarbonyl)prolinate

XLogP
0.7
TPSA (Topological Polar Surface Area)
93.2
Hydrogen Bond Donors
0
Hydrogen Bond Acceptors
6
Rotatable Bonds
5
Heavy Atoms
22
Complexity
494.0
Exact Mass
312.13214
Monoisotopic Mass
312.13214
Data Source: Chemical property values are referenced from PubChem, the world's largest open chemistry database maintained by the National Center for Biotechnology Information (NCBI), U.S. National Library of Medicine.

Property Insights of 2,5-Dioxopyrrolidin-1-yl 1-(tert-butoxycarbonyl)prolinate

The XLogP value of 0.7 suggests moderate lipophilicity, balancing water solubility and membrane permeability for 2,5-Dioxopyrrolidin-1-yl 1-(tert-butoxycarbonyl)prolinate. The TPSA of 93.2 Ų falls within the moderate polarity range, balancing permeability and solubility for 2,5-Dioxopyrrolidin-1-yl 1-(tert-butoxycarbonyl)prolinate. Following Lipinski's Rule of Five, 2,5-Dioxopyrrolidin-1-yl 1-(tert-butoxycarbonyl)prolinate has 0 hydrogen bond donor(s) and 6 hydrogen bond acceptor(s), all within the drug-like range, suggesting favorable oral bioavailability potential.

Frequently Asked Questions

What is the typical lead time for this product?
Lead time typically ranges from 3-7 business days for in-stock items. For larger quantities or custom orders, please contact us for specific lead times.
Can you provide samples for testing?
Yes, we offer sample quantities for quality testing. Please submit an inquiry with your requirements and we will arrange samples accordingly.
What documentation do you provide with the product?
We provide COA (Certificate of Analysis), MSDS (Material Safety Data Sheet), and technical data sheets with each shipment.
Do you ship internationally?
Yes, we ship to most countries worldwide. Shipping costs and delivery times vary by location. Please contact us for specific shipping information.

Frequently Asked Questions

What is the CAS number of 2,5-Dioxopyrrolidin-1-yl 1-(tert-butoxycarbonyl)prolinate?

The CAS number of 2,5-Dioxopyrrolidin-1-yl 1-(tert-butoxycarbonyl)prolinate is 102185-34-2.

What is the molecular formula of 2,5-Dioxopyrrolidin-1-yl 1-(tert-butoxycarbonyl)prolinate?

The molecular formula of 2,5-Dioxopyrrolidin-1-yl 1-(tert-butoxycarbonyl)prolinate is C14H20N2O6.

What is the molecular weight of 2,5-Dioxopyrrolidin-1-yl 1-(tert-butoxycarbonyl)prolinate?

The molecular weight of 2,5-Dioxopyrrolidin-1-yl 1-(tert-butoxycarbonyl)prolinate is 312.13 g/mol.

Where can I buy 2,5-Dioxopyrrolidin-1-yl 1-(tert-butoxycarbonyl)prolinate?

You can request a quote for 2,5-Dioxopyrrolidin-1-yl 1-(tert-butoxycarbonyl)prolinate directly from KEHONG BIO. Contact us or email info@kehongbio.com for pricing and availability.

Does KEHONG BIO offer custom synthesis for 2,5-Dioxopyrrolidin-1-yl 1-(tert-butoxycarbonyl)prolinate?

Yes, KEHONG BIO provides custom synthesis services for 2,5-Dioxopyrrolidin-1-yl 1-(tert-butoxycarbonyl)prolinate and related compounds. Contact us with your specific requirements including quantity, purity, and timeline.

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